SYNTHESIS OF 2,5-DIHYDROISOTHIAZOLE DERIVATIVES. 2. 3-ARYL(HETARYL)-SUBSTITUTED 2-ALKYL-5-ARYLIMINO-2,5-DIHYDROISOTHIAZOLES

Authors

  • И. Скрастиня Latvian Institute of Organic Synthesis
  • А. Баран Latvian Institute of Organic Synthesis
  • Д. Муцениеце Latvian Institute of Organic Synthesis
  • Ю. Попелис Latvian Institute of Organic Synthesis

DOI:

https://doi.org/10.1007/1457

Keywords:

2-alkyl-3-aryl(hetaryl)-5-arylimino-2, 5-dihydroisothiazole, N-arylamides of 3-alkylamino-3 aryl(hetaryl)prop-2-enethioic acid, oxidative cyclization

Abstract

A series of new 2-alkyl-5-arylimino-2,5-dihydroisothiazoles, substituted at position 3 with aryl and hetaryl groups and not substituted at position 4 was prepared by oxidative cyclization of N-arylamides of 3-alkylaminoprop-2-enethioic acids. The formation of the starting thioanilides was investigated by reacting the respective N-alkylimines of acetophenones with isothiocyanates. The main by-products were identified and characterized.

How to Cite
Skrastiņa, I.; Baran, A.; Muceniece, D.; Popelis, J. Chem. Heterocycl. Compd. 2014, 50, 87. [Khim. Geterotsikl. Soedin. 2014, 96.]

For this article in the English edition see DOI 10.1007/s10593-014-1451-1

Author Biographies

И. Скрастиня, Latvian Institute of Organic Synthesis

Ингрида Скрастиня

ассистент

А. Баран, Latvian Institute of Organic Synthesis

Андрей Баран

научный сотрудник

Д. Муцениеце, Latvian Institute of Organic Synthesis

Дзинтра Муцениеце

ведущий научный сотрудник

Ю. Попелис, Latvian Institute of Organic Synthesis

Юрис Попелис

ведущий научный сотрудник

Published

2014-02-10

Issue

Section

Original Papers