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SYNTHESIS OF N-ALKYLATED BENZO- AND PYRIDOTHIENOPYRROLO[1,2-a][1,4]DIAZEPIN-6-ONES ACTING AS ANTIDOTES AGAINST THE HERBICIDE 2,4-D

Татьяна А. Строганова, Владимир К. Василин, Геннадий Д. Крапивин, Владимир Д. Стрелков, Людмила В. Дядюченко
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Abstract


We report N-alkylation reactions of pyrrolo[1,2-a][1,4]diazepin-6-ones annelated with a benzene ring or thieno[2,3-b]pyridine system. A range of new N5-substituted pyrrolodiazepines were synthesized, including compounds acting as antidotes against the herbicide 2,4-D.

How to Cite
Stroganova, T. A.; Vasilin, V. K.; Krapivin, G. D.; Strelkov, V. D.; Dyadyuchenko, L. V. Chem. Heterocycl. Compd. 2016, 52, 45. [Khim. Geterotsikl. Soedin. 2016, 52, 45.]

For this article in the English edition see DOI 10.1007/s10593-016-1830-x


Keywords


annelated pyrrolo[1,2-a][1,4]diazepinones; N-alkylation; antidotes; biological activity; herbicide 2,4-D

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