1,2,3,4-TETRAHYDROPYRIMIDO[1,2-a]BENZIMIDAZOL-2- AND -4-ONES

В. B. Липсон, В. Д. Орлов, С. М. Десенко, C. В. Шишкина, O. B. Шишкин, М. Г. Широбокова

Abstract


We have studied the reaction of 2-aminobenzimidazole with esters of substituted cinnamic acids and arylidene derivatives of Meldrum's acid, and have established the direction of formation of the tetrahydrooxopyrimidine ring. We have conducted an X-ray diffraction study of 2-phenyl-1,2,3,4-tetrahydropyrimido[1,2-a]benzimidazol-4-one.

Authors: V. V. Lipson, V. D. Orlov, S. M. Desenko, S. V. Shishkina, O. V. Shishkin, and M. G. Shirobokova.

English Translation in Chemistry of Heterocyclic Compounds, 2000, 36 (9), pp 1039-1043

http://link.springer.com/article/10.1023/A%3A1002777714158


Keywords


2-aminobenzimidazole; arylidene derivatives of Meldrum's acid; partially hydrogenated pyrimido[1,2-a]benzimidazoles; esters of substituted cinnamic acids; X-ray diffraction study; ring condensation

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