FORMYLATION OF 3,4-DIHYDROPYRROLO[1,2-<i>a</i>]PYRAZINES

Authors

  • В. И. Теренин M. V. Lomonosov Moscow State University
  • Н. А. Целищева M. V. Lomonosov Moscow State University
  • E. B. Kабанова M. V. Lomonosov Moscow State University
  • А. П. Плешкова M. V. Lomonosov Moscow State University
  • Н. B. Зык M. V. Lomonosov Moscow State University

DOI:

https://doi.org/10.1007/369

Keywords:

3, 4-dihydropyrrolo[1, 2-a]pyrazine, Vilsmeier formylation

Abstract

Formylation of 3,4-dihydropyrrolo[1,2-a]pyrazines containing alkyl or aryl substituents at position 1 has been studied under the conditions of the Vilsmeier reaction. The direction of the reaction depends on the structure of 3,4-dihydropyrrolo[1,2-a]pyrazine starting materials. Formylation of 1-methyl-substituted 3,4-dihydropyrrolo[1,2-a]pyrazines occurs at the methyl group.

Authors: V. I. Terenin, N. A. Tselishcheva, E. V. Kabanova, A. P. Pleshkova, and N. V. Zyk.

English Translation in Chemistry of Heterocyclic Compounds, 2000, 36 (10), pp 1206-1212

http://link.springer.com/article/10.1023/A%3A1002876901829

Published

2013-03-05

Issue

Section

Original Papers