METHYL TRIFLUOROPYRUVATE <i>N</i>-(PYRIMIDIN-2-YL)IMINES IN CYCLOCONDENSATION REACTIONS WITH 1,3-BINUCLEOPHILIC REAGENTS

Authors

  • В. Б. Соколов Институт физиологически активных веществ РАН
  • А. Ю. Аксиненко Институт физиологически активных веществ РАН
  • Т. А. Епишина Институт физиологически активных веществ РАН
  • Т. В. Горева Институт физиологически активных веществ РАН

DOI:

https://doi.org/10.1007/467

Keywords:

2-aminothiazoline, 6-aminouracils, N-benzylbenzamidine, 3, 5-dihydroimidazol-4-ones, 2, 3 dihydroimidazo[2, 1-d][1, 3]thiazol-5(6H)-one, 4, 5-dihydro-1H-pyrroles, 5, 7-dihydro-1H-pyrrolo[2, 3-d]- pyrimidine-2, 6-triones, imidazolidine-2, 4-dione, methyl 3-aminocrotonate, methyl trifluoropyruvate N (pyrimidin-2-yl)imines, N-substituted ureas, cyclocondensation

Abstract

Cyclocondensation reactions of methyl trifluoropyruvate N-(pyrimidin-2-yl)imines with N-substituted ureas, N-benzylbenzamidine, 2-aminothiazoline, methyl 3-aminocrotonate, and 6-aminouracils leading to imidazolidine-2,4-diones, 3,5-dihydroimidazol-4-ones, 2,3-dihydroimidazo[2,1-d][1,3]thiazol-5(6H)-one, 4,5-dihydro-1H-pyrroles, and 5,7-dihydro-1H-pyrrolo[2,3-d]pyrimidine-2,4,6-triones have been studied.

Authors: V. B. Sokolov, A. Yu. Aksinenko, T. A. Epishina, and T. V. Goreva

English Translation in Chemistry of Heterocyclic Compounds, 2013, 49 (3), pp 435-439

http://link.springer.com/article/10.1007/s10593-013-1265-6

Downloads

Published

2013-04-05

Issue

No. 3 (2013)

Section

Original Papers