

CYCLOPROPYLATION OF HETEROCYCLIC CORES USING CYCLOPROPYLBORONIC DERIVATIVES

Abstract
Methods for cyclopropane ring incorporation into various heterocyclic cores using cyclopropylsubstituted organoboron compounds are surveyed. In particular, Suzuki–Miyaura and Chan–Lam reactions, recent coupling processes involving organotrifluoroborates, as well as C–H activation of
heterocyclic substrates are discussed.
heterocyclic substrates are discussed.
Keywords
organoboron compounds; cyclopropane; coupling reactions; nitrogen-containing heterocycles
Latvian Institute of Organic Synthesis - Aizkraukles iela, 21, Riga, LV-1006, Latvia - hgs@osi.lv