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SYNTHESIS OF NOVEL 2-HETARYLPYRROLIDINES VIA THE REACTION OF N-(4,4-DIETHOXYBUTYL)AMIDOPHOSPHATES WITH C-NUCLEOPHILES

Андрей В. Смолобочкин, Рахымжан А. Турманов, Альмир С. Газизов, Елизавета А. Кузнецова, Александр Р. Бурилов, Михаил А. Пудовик
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Abstract


The reactions of N-(4,4-diethoxybutyl)amidophosphates with С-nucleophiles in chloroform in the presence of trifluoroacetic acid provided new 2-hetarylpyrrolidines. The reaction proceeded under mild conditions and gave good yields in the absence of metal-based catalysts.

Keywords


N-(4,4-diethoxybutyl)amidophosphate; 2-hetarylpyrrolidines; trifluoroacetic acid; heterocyclization.

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