

SYNTHESIS OF NOVEL 2-HETARYLPYRROLIDINES VIA THE REACTION OF N-(4,4-DIETHOXYBUTYL)AMIDOPHOSPHATES WITH C-NUCLEOPHILES

Abstract
The reactions of N-(4,4-diethoxybutyl)amidophosphates with С-nucleophiles in chloroform in the presence of trifluoroacetic acid provided new 2-hetarylpyrrolidines. The reaction proceeded under mild conditions and gave good yields in the absence of metal-based catalysts.
Keywords
N-(4,4-diethoxybutyl)amidophosphate; 2-hetarylpyrrolidines; trifluoroacetic acid; heterocyclization.
Latvian Institute of Organic Synthesis - Aizkraukles iela, 21, Riga, LV-1006, Latvia - hgs@osi.lv