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SNH AMIDATION OF 5(6,7,8)-NITROQUINOLINE N-OXIDES

Анастасия A. Боровлева, Елена K. Авакян, Гульминат A. Амангазиева, Олег П. Демидов, Диана Ю. Побединская, Артём П. Ермоленко, Александр Н. Ларин, Иван В. Боровлев
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Abstract


Direct SNH amidation of 6- and 7-nitroquinoline N-oxides in anhydrous DMSO allowed to obtain N-oxides of 2- and 8-aroylaminonitroquinolines, respectively. 5-Nitroquinoline N-oxide was transformed into a mixture of amides derived from the N-oxides of 5-nitro and 5-nitrosoquinolines. 8-Nitroquinoline N-oxide underwent destruction under the same conditions.

Keywords


N-(nitro(nitroso)-1-oxidoquinolinyl)benzamides; 5(6,7,8)-nitroquinoline N-oxides; SNH amidation; disproportionation.

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