CHEMISTRY OF 3-ACYL-2-HALOINDOLES

Authors

  • С. В. Денькина Scientific Research Institute of Physical and Organic Chemistry, Southern Federal University
  • К. Ф. Суздалев Scientific Research Institute of Physical and Organic Chemistry, Southern Federal University

DOI:

https://doi.org/10.1007/873

Keywords:

aldehyde, 3-acyl-2-haloindoles, indole, [a]-fused indoles, [b]-fused indoles

Abstract

Methods for the synthesis and transformation of 3-acyl-2-haloindoles, which are polyfunctional reagents used for preparing various indole derivatives, are summarized. The reduction and oxidation of the acyl group, condensation at the carbonyl group, nucleophilic and radical substitution of the halogen atom are considered. Reactions leading to [b]-fused indoles are discussed separately.

Authors: S. V. Den'kina and K. F. Suzdalev

English Translation in Chemistry of Heterocyclic Compounds, 2012, 48 (11), pp 1581-1612

http://link.springer.com/article/10.1007/s10593-013-1181-9

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Published

2013-08-22

Issue

No. 11 (2012)

Section

Review Articles