

2018 No. 12 (618) pp. 1083-1174
Table of Contents
Anniversaries and dates
PROFESSOR ALEKSANDER FEDOROVICH POZHARSKII. TO THE 80TH BIRTHDAY |
PDF (Russian)
![]() |
1083 |
Review Articles
1,3-DIPOLAR CYCLOADDITION REACTIONS OF AZOMETHINE YLIDES AND ALKYNES |
PDF (Russian)
![]() |
Анна В. Гулевская, Юлия И. Нелина-Немцева | 1084-1107 |

Heterocycles in Focus
TETRAHYDRO-4H-THIOPYRAN-4-ONE IN MULTICOMPONENT REACTIONS (MICROREVIEW) |
PDF (Russian)
![]() |
Лариса А. Баева | 1108-1110 |

Original Papers
FACILE ONE-POT SYNTHESIS OF N-FUSED 1,2,4-TRIAZOLES via OXIDATIVE CYCLIZATION USING MANGANESE DIOXIDE |
PDF
![]() |
Ashish Bhatt, Rajesh K. Singh, Ravi Kant | 1111-1116 |

1,3-DIPOLAR CYCLOADDITION OF DIPHENYLNITRILIMINE AND 5-ARYLMETHYLIDENE-1-PHENYL-1,5,6,7-TETRAHYDRO-4H-INDAZOL-4-ONES TO AFFORD NOVEL SPIRO[INDAZOLE-5,3'-PYRAZOLE] DERIVATIVES |
PDF
![]() |
Ren Demin, Kuang Guojiang, Li Xiaofang | 1117-11120 |

SYNTHESIS OF β-(o-HYDROXYBENZYL)PYRIDINES BY THREE-COMPONENT CONDENSATION OF AMMONIA, CARBONYL-SUBSTITUTED 4Н-CHROMENES, AND СН ACIDS |
PDF (Russian)
![]() |
Дмитрий В. Осипов, Виталий А. Осянин, Юрий Н. Климочкин | 1121-1126 |

MULTICOMPONENT SYNTHESIS OF UNSYMMETRICAL 5-NITROPYRIDINES |
PDF (Russian)
![]() |
Владислав A. Ковеза, Иван B. Кулаков, Зарина T. Шульгау, Тулеген M. Сейлханов | 1127-1130 |

SYNTHESIS OF HYBRID MOLECULES CONTAINING PYRIMIDINE AND DITERPENE ALKALOID LAPPACONITINE FRAGMENTS |
PDF (Russian)
![]() |
Эльвира Э. Шульц, Кирилл П. Черемных, Виктор А. Савельев, Олег П. Шкурко | 1131-1138 |

NEW SPIRO DERIVATIVE OF DIHYDRO-1,2,3-TRIAZOLO[1,5-a]PYRIMIDINE AS A PRODUCT OF MULTICOMPONENT REACTION |
PDF
![]() |
Eugene S. Gladkov, Svetlana M. Sirko, Vladimir I. Musatov, Svetlana V. Shishkina, Irina G. Tkachenko, Sergey A. Komykhov, Sergey M. Desenko | 1139-1144 |

SYNTHESIS AND PROPERTIES OF 5-ARYL-3-DIAZO-3H-PYRAZOLES AND 3-ARYL-1H-PYRAZOLE-5-DIAZONIUM SALTS. PREPARATION AND CYTOLYTIC ACTIVITY STUDIES OF 2-ARYLPYRAZOLO- [5,1-c][1,2,4]BENZOTRIAZINES |
PDF (Russian)
![]() |
Дарья Л. Алексеева, Виктория Ю. Рахимова, Артем С. Минин, Анна В. Белоусова, Елена В. Садчикова | 1145-1152 |

AN EFFICIENT METHOD FOR THE SYNTHESIS OF 2-THIAZOLEACETIC ACID N-SULFONYL AMIDINES |
PDF (Russian)
![]() |
Владимир Г. Илькин, Василий А. Бакулев, Вера С. Берсенева, Павел А. Слепухин | 1153-1160 |

MICROWAVE-ASSISTED CU-CATALYZED C–C BOND FORMATION: ONE-POT SYNTHESIS OF FULLY SUBSTITUTED 1,2,3-TRIAZOLES USING NONSYMMETRICAL IODOALKYNES AND THEIR BIOLOGICAL EVALUATION |
PDF
![]() |
Nagavelli Vasudeva Reddy, Sirassu Narsimha, Kumaraswamy Battula, Yellu Narsimha Reddy | 1161-1167 |

Short Communications
THE POTENTIAL OF EMPLOYING SUBSTITUTED BIS[3-HYDROXY-2-(PYRIMIDIN-2-YL)-2Н-PYRAZOL-4-YL]METHANE FOR THE SYNTHESIS OF SYMMETRICAL N,O-MACROHETEROCYCLES WITH A DIOXACYCLOALKANE CENTRAL FRAGMENT |
PDF (Russian)
![]() |
Андрей В. Еркин, Владислав В. Гуржий, Виктор И. Крутиков | 1168-1170 |

THE INFLUENCE OF LEWIS ACID CATALYST ON THE KINETIC AND MOLECULAR MECHANISM OF NITROUS ACID ELIMINATION FROM 5-NITRO-3-PHENYL-4,5-DIHYDROISOXAZOLE: DFT COMPUTATIONAL STUDY |
PDF
![]() |
Agnieszka Łapczuk-Krygier, Jolanta Jaśkowska, Radomir Jasiński | 1172-1174 |

Latvian Institute of Organic Synthesis - Aizkraukles iela, 21, Riga, LV-1006, Latvia - hgs@osi.lv