Vol 56, No 6 (2020)

Heterocyclic Compounds in Medicinal Chemistry

Open Access Open Access  Restricted Access Subscription Access
2020 No.6 (636) pp. 625–804

Table of Contents

Editorial

THEMATIC ISSUE ''HETEROCYCLIC COMPOUNDS IN MEDICINAL CHEMISTRY'' PDF (Russian)
Андрей Е. Щекотихин 625

Review Articles

HETEROCYCLIC INHIBITORS OF VIROPORINS IN THE DESIGN OF ANTIVIRAL COMPOUNDS PDF (Russian)
Вадим А. Ширяев, Юрий Н. Климочкин 626-635
NUCLEOSIDE ANALOGS WITH FLEXIMER NUCLEOBASE PDF (Russian)
Михаил В. Чудинов 636-643
INDOLO[2,3-a]CARBAZOLES: DIVERSITY, BIOLOGICAL PROPERTIES, APPLICATION IN ANTITUMOR THERAPY PDF (Russian)
Роман Г. Зенков, Лидия В. Эктова, Ольга А. Власова, Геннадий А. Белицкий, Марианна Г. Якубовская, Кирилл И. Кирсанов 644-658
FAVIPIRAVIR – A MODERN ANTIVIRAL DRUG: SYNTHESIS AND MODIFICATIONS PDF (Russian)
Юлия А. Титова, Ольга В. Федорова 659-662
IMIDAZO[a]QUINOXALINES: NEW APPROACHES TO SYNTHESIS AND BIOLOGICAL ACTIVITY PDF (Russian)
Алексей А. Калинин, Лилия H. Исламова, Гузель M. Фазлеева 663-673
DIAZAPYRENES: INTERACTION WITH NUCLEIC ACIDS AND BIOLOGICAL ACTIVITY PDF (Russian)
Андрей М. Жиров, Дмитрий А. Ковалев, Диана В. Ульшина, Сергей В. Писаренко, Олег П. Демидов, Иван В. Боровлев 674-693
THE MAIN DIRECTIONS AND RECENT TRENDS IN THE SYNTHESIS AND USE OF ISOXAZOLES PDF (Russian)
Оксана Б. Бондаренко, Николай В. Зык 694-707
SYNTHESIS AND BIOLOGICAL ACTIVITIES OF 4H-3,1-BENZOTHIAZIN-4-ONES PDF
Lan Phuong Vu, Michael Gütschow 708-714
OXABORINE DERIVATIVES: SYNTHESIS AND THERAPEUTIC POTENTIAL PDF (Russian)
Анна Н. Тевяшова 715-718

Heterocycles in Focus

PHOTOREGULATED MACROCYCLIC CELL-PENETRATING PEPTIDES PDF
Igor V. Komarov, Iuliia V. Bakanovych 719-721

Original Papers

ION EXCHANGE RESIN-CATALYZED SYNTHESIS OF BRIDGED TETRAOXANES POSSESSING IN VITRO CYTOTOXICITY AGAINST HELA CANCER CELLS PDF
Vera A. Vil', Ivan A. Yaremenko, Dmitri I. Fomenkov, Dmitri O. Levitsky, Fabrice Fleury, Alexander O. Terent'ev 722-726
HETEROCYCLIC ANALOGS OF 5,12-NAPHTHACENEQUINONE 16*. SYNTHESIS AND PROPERTIES OF NEW DNA LIGANDS BASED ON 4,11-DIAMINOANTHRA[2,3-b]THIOPHENE-5,10-DIONE PDF (Russian)
Дарья B. Андреева, Александр С. Тихомиров, Любовь Г. Деженкова, Дмитрий Н. Калюжный, Ольга К. Мамаева, Светлана Е. Соловьева, Юрий Б. Синькевич, Андрей Е. Щекотихин 727-733
SYNTHESIS AND ANTIPROLIFERATIVE ACTIVITY OF SALICYLIDENEHYDRAZONES BASED ON INDOLE-2(3)-CARBOXYLIC ACIDS PDF (Russian)
Андрей Г. Васин, Любовь Г. Деженкова, Иван В. Иванов, Александр М. Щербаков, Андрей Е. Щекотихин 734-740
SYNTHESIS AND STUDY OF CYTOTOXIC ACTIVITY OF NOVEL 3,3-BIS(INDOL-3-YL)-1,3-DIHYDROINDOL-2-ONES PDF (Russian)
Сергей Н. Лавренов, Ольга П. Бычкова, Любовь Г. Деженкова, Артур С. Мкртчян, Виктор В. Татарский, Елена А. Цвигун, Алексей С. Тренин 741-746
SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL DISPIRO COMPOUNDS BASED ON 5-ARYLIDENEHYDANTOINS AND ISATINS AS INHIBITORS OF P53–MDM2 PROTEIN–PROTEIN INTERACTION PDF
Anastasia Beloglazkina, Alexander Barashkin, Vladislav Polyakov, German Kotovsky, Nikita Karpov, Sofia Mefedova, Bogdan Zagribelny, Yan Ivanenkov, Marina Kalinina, Dmitry Skvortsov, Victor Tafeenko, Nikolay Zyk, Alexander Majouga, Elena Beloglazkina 747-755
STRUCTURE AND ANTIBACTERIAL ACTIVITY (MEDIATED BY THE SOS RESPONSE) OF SPIROPIPERIDINIUM SALTS OBTAINED BY CYCLIZATION OF MANNICH BASES OF ARYLALIPHATIC 1,5-DIKETONES PDF (Russian)
Алексей В. Букреев, Таисия И. Акимова, Илья А. Остерман, Анна Н. Шахтина, Юлия В. Худякова, Андрей В. Герасименко, Петр В. Сергиев, Ольга А. Донцова, Павел И. Дерябин, Вера Б. Колычева 756-762
SYNTHESIS OF CYCLIC D-(+)-CAMPHORIC ACID IMIDES AND STUDY OF THEIR ANTIVIRAL ACTIVITY PDF
Vladimir V. Chernyshov, Olga I. Yarovaya, Roman Yu. Peshkov, Nariman F. Salakhutdinov 763-768
THE SYNTHESIS OF NEW ACYCLIC ANALOGS OF 3-PHENACYLURIDINE AND COMPARATIVE EVALUATION OF THEIR IN VIVO BIOLOGICAL ACTIVITY PDF (Russian)
Иван А. Новаков, Лейла Л. Брунилина, Иван А. Кириллов, Максим Б. Навроцкий, Мария Д. Робинович, Евгения С. Титова, Дмитрий С. Шейкин, Евсей А. Ручко, Алла В. Павлова, Анастасия А. Котлярова, Татьяна Г. Толстикова 769-775
8-ETHYNYLXANTHINES AS PROMISING ANTIPROLIFERATIVE AGENTS, ANGIOGENESIS INHIBITORS, AND CALCIUM CHANNEL ACTIVITY MODULATORS PDF
Pavel Arsenyan, Jelena Vasiljeva, Ilona Domracheva, Iveta Kanepe-Lapsa 776-785
SYNTHESIS OF 2-AMINOPYRIDOPYRIMIDINONES AND THEIR PLASMEPSIN I, II, IV INHIBITION POTENCY PDF
Dace Rasina, Georgijs Stakanovs, Iveta Kanepe-Lapsa, Raitis Bobrovs, Kristaps Jaudzems, Aigars Jirgensons 786-792
CAGE-LIKE AMINES IN THE GREEN PROTOCOL OF TRANSANNULAR THIENO[2,3-d]PYRIMIDINONE FORMATION AS PROMISING ANTICANCER AGENTS PDF
Olga Ya. Shyyka, Nazariy T. Pokhodylo, Vitalii A. Palchykov, Nataliya S. Finiuk, Rostyslav S. Stoika, Mykola D. Obushak 793-799

Short Communications

INDOLE DERIVATIVES OF FUSIDANE TRITERPENOIDS: SYNTHESIS AND THE ANTIBACTERIAL ACTIVITY PDF (Russian)
Елена Е. Салимова, Айгуль А. Магафурова, Елена В. Третьякова, Ольга С. Куковинец, Людмила В. Парфенова 800-804


 

 

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