Vol 57, No 11 (2021)

Open Access Open Access  Restricted Access Subscription Access
2021 № 11 (653) p. 1061–1148

Table of Contents

Review Articles

PYRAZOLES, ISOXAZOLES, AND 1,2,3-TRIAZOLES AS ANALOGS OF THE NATURAL CYTOSTATIC COMBRETASTATIN A-4: EFFICIENT ROUTES OF SYNTHESIS, TUBULIN INHIBITION, AND CYTOTOXICITY PDF (Russian)
Роман К. Костин, Александр С. Маршавин 1061-1072

Heterocycles in Focus

SYNTHESIS OF 2H-THIOCHROMENE DERIVATIVES PDF
Seyed Sajad Sajadikhah, Mahmoud Nassiri 1073-1075
SYNTHESIS OF HETEROCYCLIC RING-FUSED QUINONES PDF
Anastasija Gaile, Nelli Batenko 1076-1078

Original Papers

REACTIVITY OF ALICYCLIC 1,5,9-TRIKETONES TOWARD FIVE-, SIX-, AND SEVEN-MEMBERED RINGS IN ACIDIC MEDIUM. STEREOCHEMISTRY OF INTRAMOLECULAR CYCLIZATION PRODUCTS PDF (Russian)
Таисия И. Акимова, Ольга А. Солдаткина, Андрей В. Герасименко, Вячеслав Г. Савченко, Алевтина А. Капустина 1079-1085
AZIRIDINE-2-CARBOXYLIC ACID DERIVATIVES AND ITS OPEN-RING ISOMERS AS A NOVEL PDIA1 INHIBITORS PDF
Irena Leite, Victor Andrianov, Diana Zelencova-Gopejenko, Einars Loza, Iveta Kazhoka-Lapsa, Ilona Domracheva, Marta Stojak, Stefan Chlopicki, Ivars Kalvins 1086-1106
[3+2] CYCLOADDITION REACTIONS OF 1-SUBSTITUTED 3,3,3-TRIFLUOROPROPENES WITH DIAZO COMPOUNDS AND NITRILIMINES – SYNTHESIS OF PYRAZOLINES AND PYRAZOLES PDF (Russian)
Юрий Н. Маркитанов, Вадим М. Тимошенко, Сергей С. Михайличенко, Эдуард Б. Русанов, Александр И. Хижан, Юрий Г. Шермолович 1107-1115
SYNTHETIC TRANSFORMATIONS OF SESQUITERPENE LACTONES. CONTROLLABLE SYNTHESIS OF 11,13-DIHYDROISOALANTOLACTONE AZIDES AND 13-(1,2,3-TRIAZOLYL)EUDESMANOLIDES BASED ON SESQUITERPENE LACTONES PDF (Russian)
Сергей С. Патрушев, Татьяна В. Рыбалова, Эльвира Э. Шульц 1116-1129
LEWIS ACID CATALYZED CONDENSATION OF 2-AMINOHETARENE N-OXIDES WITH N,N-DIMETHYLFORMAMIDE DIMETHYL ACETAL PDF (Russian)
Сергей А. Каралаш, Дмитрий М. Быстров, Иван В. Ананьев, Леонид Л. Ферштат 1130-1136
SYNTHESIS OF METHYL(ETHYL) PYRAZOLO[4,3-b]PYRIDINE-6-CARBOXYLATES AND THEIR CONVERSION TO tert-BUTYL 4,5,6,7-TETRAHYDROPYRAZOLO-[4,3-b]PYRIDINE-6-CARBOXYLATES PDF (Russian)
Георгий Г. Яковенко, Леся Н. Салиева, Эдуард Б. Русанов, Илья С. Дончак, Михаил В. Вовк 1137-1145

Short Communications

SYNTHESIS AND PERMETHYLATION OF METHYL 5-(2-CHLOROPYRIDIN-3-YL)PENTANOATES PDF
Franziska Bendrath, Peter Langer 1146-1148


 

 

Latvian Institute of Organic Synthesis - Aizkraukles iela, 21, Riga, LV-1006, Latvia - hgs@osi.lv

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