N-arylation of 1-aminobenzimidazole
Abstract
By treatment of the sodium (potassium) salt of 1-formylaminobenzimidazole in acetone or DMF with picryl chloride. 2,4-dinitrochlorobenzene, 2- and 4-nitrochlorobenzenes, we obtained the corresponding 1-aryl-aminobenzimidazoles. This is the first case of direct arylation of the amino group in N-aminobenzimidazole.
How to Cite
Pozharskii, A. F.; Dyablo, O. V.; Kuz'menko, V. V.; Evgrafova, E. A. Chem. Heterocycl. Compd. 1996, 32, 1156. [Khim. Geterotsikl. Soedin. 1996, 1347.]
For this article in the English edition, see DOI https://doi.org/10.1007/BF01169226