4-ARYL-1-HYDRAZINO-5<i>H</i>-2,3-BENZODIAZEPINE AND 1-ARYL-4-HYDRAZINO-5<i>H</i>-2,3-BENZODIAZEPINE IN THE SYNTHESIS OF CONDENSED [1,2]DIAZEPINES
DOI:
https://doi.org/10.1007/413Keywords:
[1, 2, 4]triazolo[3, 4-a][2, 3]benzodiazepine, 4]triazolo[4, 3-c][2, cyclizationAbstract
A method has been developed for the cyclization of 4-aryl-1-hydrazino-5H-2,3-benzodiazepine and 1-aryl-4-hydrazino-5H-2,3-benzodiazepine into 3-R-6-aryl-7H-[1,2,4]triazolo[3,4-a]- and 3-R-6-aryl-7H-[1,2,4]triazolo[4,3-c]benzodiazepine derivatives with various substituents in the triazole ring.
Authors: O. I. Kharaneko, V. Yu. Popov, and S. L. Bogza
English Translation in Chemistry of Heterocyclic Compounds, 2013, 49 (2), pp 317-324