EFFICIENT ONE-STEP SYNTHESIS OF 3-ARYL-2-PYRIDONES FROM 6-ARYL-1,2,4-TRIAZIN-5-ONES

Authors

  • Мария И. Савчук Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia
  • Ярослав К. Штайц Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia
  • Дмитрий С. Копчук Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 21 S. Kovalevskoi /20 Akademicheskaya St., Yekaterinburg 620219, Russia
  • Григорий В. Зырянов Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 21 S. Kovalevskoi /20 Akademicheskaya St., Yekaterinburg 620219, Russia
  • Олег С. Ельцов Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia
  • Татьяна А. Поспелова Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia
  • Владимир Л. Русинов Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 21 S. Kovalevskoi /20 Akademicheskaya St., Yekaterinburg 620219, Russia
  • Олег Н. Чупахин Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 21 S. Kovalevskoi /20 Akademicheskaya St., Yekaterinburg 620219, Russia

DOI:

https://doi.org/10.1007/5115

Keywords:

2, 2'-bipyridine, 2-pyridone, 1, 4-triazin-5-one, autoclave, aza-Diels–Alder reaction, nucleophilic ipso-substitution.

Abstract

An efficient method for the synthesis of substituted 2-pyridones based on the aza-Diels–Alder reaction of 1,2,4-triazin-5-ones and dienophiles, 2,5-norbornadiene and 4-(cyclopent-1-en-1-yl)morpholine, is proposed.

Author Biographies

Мария И. Савчук, Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia

Младший научный сотрудник, Уральский Федеральный Университет

Ярослав К. Штайц, Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia

Младший научный сотрудник, Уральский Федеральный Университет

Дмитрий С. Копчук, Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 21 S. Kovalevskoi /20 Akademicheskaya St., Yekaterinburg 620219, Russia

научный сотрудник, Группа координационных соединений

Григорий В. Зырянов, Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 21 S. Kovalevskoi /20 Akademicheskaya St., Yekaterinburg 620219, Russia

cтарший научный сотрудник, Группа координационных соединений

Олег С. Ельцов, Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia

Доцент, Уральский Федеральный Университет

Татьяна А. Поспелова, Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia

Доцент, Уральский Федеральный Университет

Владимир Л. Русинов, Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 21 S. Kovalevskoi /20 Akademicheskaya St., Yekaterinburg 620219, Russia

Зав. кафедрой ОиБХ, Уральский Федеральный Университет

Олег Н. Чупахин, Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 21 S. Kovalevskoi /20 Akademicheskaya St., Yekaterinburg 620219, Russia

Научный Руководитель

Институт Органического Синтеза, Уральское Отделение РАН, Россия, 620219, г. Екатеринбург, ул. Софьи Ковалевской, 22

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Published

2019-09-27

Issue

Vol. 55 No. 10 (2019)

Section

Original Papers