SYNTHESIS OF 2-PHENYLINDOLE N-DERIVATIVES UNDER CONDITIONS OF CATALYSIS BY PALLADIUM COMPLEXES
DOI:
https://doi.org/10.1007/528Abstract
The synthesis of 2-phenylindole N-derivatives was accomplished. The synthesis included the catalytic coupling of o-iodoaniline with phenylacetylene leading to 2-aminotolan, the preparation of the derivative of the last at the nitrogen atom, and its catalytic cyclization to the corresponding indole.
Authors: A. I. Roshchin and N. A. Bumagin.
English Translation in Chemistry of Heterocyclic Compounds, 1999, 35 (2), pp 171-175
http://link.springer.com/article/10.1007/BF02251704