SYNTHESIS AND REACTIONS OF THIOAMIDES OF 5-AMINO-2-ARYL-2H-1,2,3-TRIAZOLE-4-CARBOXYLIC ACID

Authors

  • Н. П. Бельская Ural State Technological University named of the First President of Russia B. N. Yeltsin, Ekaterinburg 620002
  • С. Г. Сапожникова Ural State Technological University named of the First President of Russia B. N. Yeltsin, Ekaterinburg 620002
  • В. А. Бакулев Ural State Technological University named of the First President of Russia B. N. Yeltsin, Ekaterinburg 620002
  • О. С. Ельцов Ural State Technological University named of the First President of Russia B. N. Yeltsin, Ekaterinburg 620002
  • П. А. Слепухин I. Ya. Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, Ekaterinburg 620041
  • Д. Фан State Key Laboratory of Elemento-Organic Chemistry, Nankai University, Tianjin, 300071

DOI:

https://doi.org/10.1007/6651

Keywords:

aminoimidazoles, α-halo ketones, thiazoles, thioamides, thioimidinium salts, 1, 2, 3-triazoles, 4-triazoles

Abstract

A method has been developed for obtaining thioamides of 5-amino-2-aryl-2H-1,2,3-triazole-4-carboxylic acid. Their heterocyclization reactions with bifunctional reagents has been studied. New heterocyclic polycyclic ensembles have been synthesized containing a 1,2,3-triazole fragment, a thiazole, and a residue of the natural alkaloid cytisine.

How to Cite
Belskaya, N. P.; Sapozhnikova, S. G.; Bakulev, V. A.; Eltsov, O. S.; Slepukhin, P. A.; Fan, Z.-J.  Chem. Heterocycl. Compd. 2009, 45, 844. [Khim. Geterotsikl. Soedin. 2009, 1061.]

For this article in the English edition see DOI 10.1007/s10593-009-0348-x


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Published

2022-03-01

Issue

No. 7 (2009)

Section

Original Papers