DICHLOROACETYLAROYLMETHANES AS TWO-CARBON SYNTHONS IN THE BIGINELLI REACTION

Authors

  • В. А. Мамедов A. E. Arbuzov Institute of Organic and Physical Chemistry, Kazan' Science Center, Russian Academy of Sciences, Kazan' 420088
  • Л. В. Мустакимова A. E. Arbuzov Institute of Organic and Physical Chemistry, Kazan' Science Center, Russian Academy of Sciences, Kazan' 420088
  • А. Т. Губайдуллин A. E. Arbuzov Institute of Organic and Physical Chemistry, Kazan' Science Center, Russian Academy of Sciences, Kazan' 420088
  • С. В. Вдовина A. E. Arbuzov Institute of Organic and Physical Chemistry, Kazan' Science Center, Russian Academy of Sciences, Kazan' 420088
  • И. А. Литвинов A. E. Arbuzov Institute of Organic and Physical Chemistry, Kazan' Science Center, Russian Academy of Sciences, Kazan' 420088
  • В. С. Резник A. E. Arbuzov Institute of Organic and Physical Chemistry, Kazan' Science Center, Russian Academy of Sciences, Kazan' 420088

DOI:

https://doi.org/10.1007/7827

Keywords:

dichloromethylacetylbenzoylmethane, urea, perhydropyrimidines, Biginelli reaction, 1H NMR spectra, cyclocondensation

Abstract

Acid-catalyzed cyclocondensation in a three component system of dichloromethylacetyl-benzoylmethanes, urea, and aromatic aldehydes occurred regio- and stereoselectively to  give polyfunctional derivatives of perhydropyrimidine.

How to Cite
Mamedov,V. A.;  Mustakimova, L. V.; Gubaidullin, A. T.; Vdovina, S. V.; Litvinov, I. A.; Reznik, V. S.  Chem. Heterocycl. Compd. 2006, 42, 1229. [Khim. Geterotsikl. Soedin. 2006, 1414.]

For this article in the English edition see DOI 10.1007/s10593-006-0230-z


Published

2023-05-24

Issue

Section

Original Papers