N-AMINATION OF UNSYMMETRICALLY SUBSTITUTED PYRIMIDINES. SYNTHESIS OF ISOMERIC N-AMINOPYRIMIDONES

Authors

  • М. Б. Бодягин St. Petersburg State University, St. Petersburg 198904, Petrodvorets
  • А. Ю. Иванов St. Petersburg State University, St. Petersburg 198904, Petrodvorets
  • K. Вурст Innsbruck University, A-6020
  • Й. Г. Шантль Innsbruck University, A-6020
  • П. С. Лобанов St. Petersburg State University, St. Petersburg 198904, Petrodvorets
  • А. А. Потехин St. Petersburg State University, St. Petersburg 198904, Petrodvorets

Keywords:

O-(mesitylenesulfonyl)hydroxylamine, 4-pyrimidones, N-amination

Abstract

N-Amination of 6-amino-2-methyl-4-pyrimidone with O-(mesitylenesulfonyl)hydroxylamine leads to the 3-amino derivative. The isomeric 1,6-diamino-2-methyl-4-pyrimidone was obtained by the N-amination of the O-benzoyl derivative of the initial pyrimidone and removal of the benzoyl protection.

How to Cite
Bodyagin, M. B.; Ivanov, A. Yu.; Wurst, K.; Schantl, J. G.; Lobanov, P. S.; Potekhin, A. A. Chem. Heterocycl. Compd. 2003, 39, 195. [Khim. Geterotsikl. Soedin. 2003, 223.]

For this article in the English edition, see DOI https://doi.org/10.1023/A:1023716424186

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Published

2003-02-25

Issue

No. 2 (2003)

Section

Original Papers