CONDENSED DIAZEPINES. SYNTHESIS OF 1-R-3,4-DIHYDRO-5<i>H</i>-BENZOTHIENO[2,3-<i>d</i>][1,2]DIAZEPIN-4-ONES
DOI:
https://doi.org/10.1007/955Keywords:
2-acyl(aroyl)benzo[b]thiophene-3-acetic acids, 1-aryl-3, 4-dihydro-5H-benzothieno[2, 3-d][1, 2]diazepin-4-ones, hydrazine hydrate, cyclizationAbstract
Novel 1-R-3,4-dihydro-5H-benzothieno[2,3-d][1,2]diazepin-4-ones have been prepared by the cyclization of 2-acyl(aroyl)benzo[b]thiophene-3-acetic acids or 1-R-benzothieno[2,3-c]pyr-3-ones with hydrazine hydrate.
Authors: V. S. Tolkunov, A. B. Eres'ko, A. V. Mazepa, G. V. Palamarchuk, O. V. Shishkin, and S. V. Tolkunov
English Translation in Chemistry of Heterocyclic Compounds, 2012, 48 (9), pp 1371-1381
http://link.springer.com/article/10.1007/s10593-012-1146-4