

2019 No.2 (620) pp. 103–192
Table of Contents
Review Articles
SYNTHESIS AND PROPERTIES OF 2,3-HETEROANNULATED THIOCHROMONES – HETERO ANALOGS OF THIOXANTHONE |
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Вячеслав Я. Сосновских | 103-125 |

Heterocycles in Focus
RECENT APPLICATION OF ELEMENTAL SULFUR IN THE SYNTHESIS OF S-HETEROCYCLES |
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Mátyás Milen, Tímea Szabó | 126-128 |

Original Papers
SYNTHESIS AND PROPERTIES OF 1-[(ADAMANTAN-1-YL)METHYL]- 3-PYRAZOLYL UREAS |
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Владимир С. Дьяченко, Дмитрий В. Данилов, Татьяна К. Шкинева, Ирина А. Вацадзе, Владимир В. Бурмистров, Геннадий Михайлович Бутов | 129-134 |

SYNTHETIC MODIFICATIONS OF CARBOLINE ALKALOID HARMINE: SYNTHESIS OF 8-SUBSTITUTED DERIVATIVES |
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Сергазы М. Адекенов, Пернеш Ж. Жанымханова, Жангельды С. Нурмаганбетов, Асел Аманжан, Сергей В. Чернов, Aйбек Ж. Турмухамбетов, Ирина Ю. Багрянская, Юрий В. Гатилов, Эльвира Э. Шульц | 135-141 |

REACTIVITY OF OXIMES OF 1-ARYL(HETARYL)-2-(HYDROXYAMINO)PROPAN-1-ONES WITH ETHYL GLYOXYLATE |
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Елена Б. Николаенкова, Алексей Я. Тихонов, Станислав Ю. Грищенко | 142-146 |

A NEW FACILE METHOD FOR THE SYNTHESIS OF 3-IMIDAZOLYLPROPIONIC ACID N-OXIDES |
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Anton V. Kutasevich, Valery P. Perevalov, Vitaly S. Mityanov, Boris V. Lichitsky, Andrey N. Komogortsev, Mikhail M. Krayushkin, Tatyana Yu. Koldaeva, Vladimir S. Miroshnikov | 147-155 |

SYNTHESIS OF SUBSTITUTED IMIDAZO[1,2-a]PYRIDIN-3-YL-ACETIC ACIDS BY MULTICOMPONENT CONDENSATION OF 2-AMINOPYRIDINES WITH ARYLGLYOXALS AND MELDRUM'S ACID |
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Борис В. Личицкий, Александр Д. Третьяков, Андрей Н. Комогорцев, Виталий С. Митянов, Аркадий А. Дудинов, Михаил М. Краюшкин | 156-159 |

EFFICIENT METHOD FOR THE SYNTHESIS OF 1,3-UNSUBSTITUTED 2-IMINO-5-OXOOCTAHYDROIMIDAZO[4,5-d]IMIDAZOLIUM IODIDES BASED ON THIOGLYCOLURILS |
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Vladimir V. Baranov, Evgeniya L. Yatsenko, Elizaveta K. Melnikova, Yulia V. Nelyubina, Angelina N. Kravchenko | 160-166 |

ANNULATION OF PYRROLE RING IN 4-ACYLPYRIDINE-3,5-DICARBONITRILES IN THE PRESENCE OF AMMONIA |
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Артур А. Григорьев, Яков С. Каюков, Анастасия Л. Никифорова, Сергей В. Карпов, Екатерина С. Щегравина, Ольга В. Каюкова, Виктор А. Тафеенко | 167-171 |

SPATIAL STRUCTURE AND NONTRIVIAL STEREODYNAMICS OF TRICYCLIC PERHYDRO-1,2,4,5-TETRAZINES |
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Rafael R. Kostikov, Tatiana A. Kornilova, Alexander F. Khlebnikov, Gennady V. Shustov, Alexander Yu. Ivanov, Vitaly V. Suslonov, Nikolay V. Shesternin, Mikhail A. Kuznetsov | 172-177 |

THIAZOLIDINE-2,4-DIONE IN BENZOYLATION REACTION |
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Igor B. Levshin, Nina A. Rastorgeva, Alexey V. Kiselev, Alexandr S. Vedenkin, Sergey V. Stovbun, Andrey V. Churakov, Oleg Yu. Saveliev, Vladimir I. Polshakov | 178-183 |

EFFICIENT METHOD FOR THE SYNTHESIS OF NOVEL SUBSTITUTED THIENO[2,3-d]PYRIMIDINE-4-CARBOXYLIC ACIDS, THEIR DERIVATIZATION, AND ANTIMICROBIAL ACTIVITY |
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Елена Д. Власова, Константин Ю. Кроленко, Максим А. Нечаев, Павел Е. Шинкаренко, Владимир И. Кабачный, Сергей В. Власов | 184-188 |

Short Communications
SYNTHESIS OF 4-POLYFLUOROALKYL-1,3-DITHIOLANES via [3+2] CYCLOADDITION OF THIOCARBONYL YLIDE TO POLYFLUOROALKANETHIOAMIDES |
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Сергей С. Михайличенко, Юрий Н. Маркитанов, Тимофей В. Руденко, Эдуард Б. Русанов, Юрий Г. Шермолович | 189-192 |

Latvian Institute of Organic Synthesis - Aizkraukles iela, 21, Riga, LV-1006, Latvia - hgs@osi.lv