SYNTHESIS AND FUNGICIDAL ACTIVITY OF ALKYL(ARYL)-SUBSTITUTED 1,3,4-THIADIAZOLIDINES

Authors

  • В. Р. Ахметова Institute of Petrochemistry and Catalysis, Russian Academy of Sciences
  • Н. Н. Махмудиярова Institute of Petrochemistry and Catalysis, Russian Academy of Sciences
  • И. С. Бушмаринов A. N. Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences
  • Г. Р. Хабибуллина Institute of Petrochemistry and Catalysis, Russian Academy of Sciences
  • Н. Ф. Галимзянова Institute of Biology, Ufa Scientific Center, Russian Academy of Sciences

DOI:

https://doi.org/10.1007/839

Keywords:

aldehydes, hydrogen sulfide, substituted hydrazines, 1, 3, 4-thiadiazolidine, fungicidal activity, cyclothiomethylation

Abstract

3,3'-Methanediylbis(4-methyl-1,3,4-thiadiazolidine) has been obtained through the cyclothio-methylation of methylhydrazine, formaldehyde, and H2S. A series of 2,5-dialkyl(aryl)-3-phenyl(benzyl)-1,3,4-thiadiazolidines has been synthesized through cyclothiomethylation of phenyl(benzyl)hydrazines with aliphatic and aromatic aldehydes and H2S. The fungicidal activity of 2,5-dimethyl-3-phenyl-1,3,4-thia-diazolidine relative to Bipolaris sorokiniana and Fusarium oxysporum has been observed, so as for the water-soluble adduct of methyl iodide and 2,5-dimethyl-3-phenyl-1,3,4-thiadiazolidine relative to Bipolaris sorokiniana.

Authors: V. R. Akhmetova, N. N. Makhmudiyarova, I. S. Bushmarinov, G. R. Khabibullina, and N. F. Galimzyanova.

English Translation in Chemistry of Heterocyclic Compounds, 2013, 49 (8), pp 1224-1231

http://link.springer.com/article/10.1007/s10593-013-1366-2

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Published

2013-08-13

Issue

No. 8 (2013)

Section

Original Papers