Synthesis, alkylation, and structural studies of 2-vinylpyrrolo[1,2-<i>a</i>]indoles

Authors

  • Н. З. Тугушева Center for the Chemistry of Medicinals, All-Russian Chemico-Pharmaceutical Scientific Research Institute, Moscow 119815
  • С. Ю. Рябова Center for the Chemistry of Medicinals, All-Russian Chemico-Pharmaceutical Scientific Research Institute, Moscow 119815
  • H. П. Соловьева Center for the Chemistry of Medicinals, All-Russian Chemico-Pharmaceutical Scientific Research Institute, Moscow 119815
  • B. Г. Граник Center for the Chemistry of Medicinals, All-Russian Chemico-Pharmaceutical Scientific Research Institute, Moscow 119815

Abstract

2-Piperidinomethylene-2H-pyrrolo[l,2-a]indole-3,9-dione can readily react with substances having an active methylene unit to form piperidinium salts which are converted to 2-vinyl pyrrolo[1,2-a]indoles. They can also undergo O-methylation using dimethyl sulfate in polar and non polar solvents to form the 9-alkoxy derivatives.

How to Cite
Tugusheva, N. Z.; Ryabova, S. Y.; Solov'eva, N. P.; Granik, V. G. Chem. Heterocycl. Compd. 1994, 30, 689. [Khim. Geterotsikl. Soedin. 1994, 781.]

For this article in the English edition, see DOI https://doi.org/10.1007/BF01166309

Published

1994-06-25

Issue

Section

Original Papers