

2016 No. 11 (593) pp. 855–972
Table of Contents
Editorial
Неклассические методы активации в химии гетероциклических соединений |
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В. А. Чебанов | 855 |
Review Articles
MECHANOCHEMICAL AND SONOCHEMICAL HETEROCYCLIZATIONS |
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Emanuela Calcio Gaudino, Silvia Tagliapietra, Stefano Mantegna, Giancarlo Cravotto | 856-865 |

REACTIONS OF 3(5)-AMINOISOXAZOLES USING CLASSICAL METHODS OF ACTIVATION, MICROWAVE IRRADIATION, AND ULTRASONICATION |
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Владимир B. Ткаченко, Валентин А. Чебанов | 866-886 |

MICROWAVE ACTIVATION IN TETRAZOLE CHEMISTRY |
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Леонид В. Мызников, Светлана В. Ворона, Татьяна В. Артамонова, Юрий Э. Зевацкий | 887-893 |

Heterocycles in Focus
SYNTHESIS OF HIGHLY SUBSTITUTED 2-PYRIDONES |
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Maria A. Vodolazhenko, Nikolay Yu. Gorobets | 894-896 |

Original Papers
FISCHER INDOLE SYNTHESIS OF 3-BENZYL-1H-INDOLE VIA CONDUCTIVE AND DIELECTRIC HEATING |
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Jesco Panther, Julian Rechmann, Thomas J. J. Müller | 897-903 |

MICROWAVE-ASSISTED SYNTHESIS OF 4-(2,2'-BISTHIOPHEN-5-YL)-5-PHENYLPYRIMIDINE DERIVATIVES WITH APPLICATIONS IN SENSORS OF NITROAROMATIC EXPLOSIVES |
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Егор В. Вербицкий, Екатерина М. Чепракова, Анна А. Баранова, Константин О. Хохлов, Ксения И. Луговик, Геннадий Л. Русинов, Олег Н. Чупахин, Валерий Н. Чарушин | 904-909 |

SYNTHESIS OF (1,2,3-THIADIAZOLYL)IMIDAZOLIDINE-2,4-DIONES BY MICROWAVE IRRADIATION AND CHARACTERIZATION OF THEIR BIOLOGICAL ACTIVITY |
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Татьяна А. Калинина, Лилия А. Хамидуллина, Юлия С. Шахмина, Татьяна В. Глухарева, Алена А. Кочубей, Ольга Е. Черепанова, Жи-Джин Фан, Юджи Жу | 910-917 |


MICHAEL ADDITION TO UNPROTECTED 3-(2-NITROVINYL)INDOLES UNDER THE CONDITIONS OF MICROWAVE SYNTHESIS |
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Александр В. Аксенов, Николай А. Аксенов, Антон А. Скоморохов, Инна В. Аксенова, Георгий Д. Грязнов, Леонид Г. Воскресенский, Михаил А. Рубин | 923-927 |

SYNTHESIS OF PYRAZOLYLFURO[2,3-f]CHROMENES AND EVALUATION OF THEIR ANTIMICROBIAL ACTIVITY |
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Dongamanti Ashok, Kavitha Rangu, Srinivas Gundu, Velagapuri Hanumantha Rao | 928-933 |

HETEROCYCLIZATION REACTIONS OF 3-METHYLISOXAZOL-5-AMINE WITH PYRUVIC ACID DERIVATIVES USING CLASSICAL AND NON-CLASSICAL ACTIVATION METHODS |
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Алиса Д. Морозова, Елена А. Муравьева, Сергей М. Десенко, Владимир И. Мусатов, Дарья В. Едаменко, Валентин А. Чебанов | 934-942 |

STUDY ON THE SCALE-UP OF PHASE-TRANSFER-CATALYZED AZO COUPLING REACTIONS IN FLOW REACTORS |
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Faith Akwi, Paul Watts | 943-947 |

EFFICIENT SYNTHESIS OF BENZIMIDAZOLES CONTAINING 1,2,4-TRIAZOL-3-ONE NUCLEUS USING MICROWAVE IRRADIATION |
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Emre Menteşe, Bahittin Kahveci | 948-951 |

PREPARATION OF BENZIMIDAZOLE N-OXIDES BY A TWO-STEP CONTINUOUS FLOW PROCESS |
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Fabrizio Politano, Elba I. Buján, Nicholas E Leadbeater | 952-957 |
ULTRASONICALLY PROMOTED SYNTHESIS OF TACRINE ANALOGS IN THE PRESENCE OF TIO2 NANOTUBES |
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Nader Ghaffari Khaligh | 958-963 |

CATALYST-FREE GREEN SYNTHESIS OF NOVEL 2-AMINO-4-ARYL-3-(4-FLUOROPHENYL)-4,6,7,8-TETRAHYDROQUINOLIN-5(1H)-ONES VIA A ONE-POT FOUR-COMPONENT REACTION UNDER ULTRASONIC CONDITION |
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Santhosh Govindaraju, Sumaiya Tabassum, Riyaz Ur-Rahaman Khan, Mohamed Afzal Pasha | 964-969 |

Letters to the Editor
SYNTHESIS OF LAPPACONITINE N-OXIDE UNDER THE CONDITIONS OF MICROWAVE ACTIVATION |
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Наталья А. Панкрушина, Кымбат Б. Рахметали | 970-972 |

Latvian Institute of Organic Synthesis - Aizkraukles iela, 21, Riga, LV-1006, Latvia - hgs@osi.lv