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2017 No. 3 (597) pp. 239–380
Table of Contents
Editorial
| PRIVILEGED HETEROCYCLIC SCAFFOLDS IN CHEMICAL BIOLOGY AND DRUG DISCOVERY: SYNTHESIS AND BIOACTIVITY |
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| Cosimo D. Altomare | 239 |
Review Articles
| N-(HETERO)ARYL-2-IMIDAZOLINES: AN EMERGING PRIVILEGED MOTIF FOR CONTEMPORARY DRUG DESIGN |
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| Mikhail Krasavin | 240-255 |
| PREPARATION AND BIOLOGICAL PROPERTIES OF 2-THIO-CONTAINING PYRIMIDINES AND THEIR CONDENSED ANALOGS |
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| Oleksii Y. Voskoboynik, Oleksandra S. Kolomoets, Galina G. Berest, Inna S. Nosulenko, Yuliya V. Martynenko, Sergiy I. Kovalenko | 256-273 |
| HETEROCYCLES AS CLASSICAL AND NONCLASSICAL RING B ISOSTERS IN COMBRETASTATIN A-4 |
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| Nikolay A. Zefirov, Olga N. Zefirova | 273-280 |
| 1,5-DIARYLPYRROLES AS POTENT ANTITUBERCULAR AND ANTI-INFLAMMATORY AGENTS |
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| Giulia Venditti, Giovanna Poce, Sara Consalvi, Mariangela Biava | 281-291 |
| 2-(AZOLYL)ANILINES: METHODS OF SYNTHESIS, CYCLOCONDENSATIONS, AND BIOLOGICAL PROPERTIES |
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| Oleksii M. Antypenko, Sergiy V. Kholodnyak, Konstantin P. Schabelnyk, Lyudmyla M. Antypenko, Sergiy Ivanovich Kovalenko | 292-309 |
Heterocycles in Focus
| 3,4-DIHYDROQUINOXALIN-2-ONES: RECENT ADVANCES IN SYNTHESIS AND BIOACTIVITIES |
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| Tone Kristoffersen, Jørn H. Hansen | 310-312 |
| SYNTHESIS OF INDOLIZINIUM SALTS |
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| Anna Ivanova, Pavel Arsenyan | 313-315 |
Original Papers
| EXPLORING THE INFLUENCE OF THE SUBSTITUENT AT POSITION 4 IN A SERIES OF 3,4-DIHYDROPYRIMIDIN-2(1H)-ONE A2B ADENOSINE RECEPTOR ANTAGONISTS |
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| Abel Crespo, Abdelaziz El Maatougui, Jhonny Azuaje, Luz Escalante, María Majellaro, María I. Loza, José Brea, María I. Cadavid, Hugo Gutiérrez-de-Terán, Eddy Sotelo | 316-321 |
| FUNCTIONALIZATION OF FOUR-MEMBERED CYCLIC SULFOXIMINES BY A CONVENIENT LITHIATION/TRAPPING SEQUENCE |
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| Arianna Tota, Flavio Fanelli, Aurelia Falcicchio, Renzo Luisi, Leonardo DEGENNARO | 322-328 |
| 2-ARYLAZETINES AS LIGANDS FOR NICOTINIC ACETYLCHOLINE RECEPTORS |
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| Leonardo Degennaro, Marina Zenzola, Annunziatina Laurino, Maria Maddalena Cavalluzzi, Carlo Franchini, Solomon Habtemariam, Rosanna Matucci, Renzo Luisi, Giovanni Lentini | 329-334 |
| SYNTHESIS AND STRUCTURE OF DIHYDROBERBERINE NITROARYL DERIVATIVES – POTENTIAL LIGANDS FOR G-QUADRUPLEXES |
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| Олег Н. Буров, Сергей В. Курбатов, Михаил Е. Клецкий, Александр Д. Загребаев, Игорь Е. Михайлов | 335-340 |
| INVESTIGATION ON THE SYNTHESIS OF NEW 3-[4-(ARYLALKOXY)PHENYLETHYL]-2-THIOXO-1,3-THIAZOLIDIN-4-ONES AND THEIR BIOLOGICAL EVALUATION AGAINST CANCER CELLS |
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| Camille D. Dago, Christelle N'ta Ambeu, Wacothon K. Coulibaly, Janat A. Mamyrbekova-Bekro, Rémy Le Guével, Anne Corlu, Jean-Pierre Bazureau | 341-349 |
| SYNTHESIS OF PHENYLPYRIDINE DERIVATIVES AND THEIR BIOLOGICAL EVALUATION TOWARD DIPEPTIDYL PEPTIDASE-4 |
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| Yan Zhu, Xiangguo Meng, Zhengyan Cai, Qun Hao, Weicheng Zhou | 350-356 |
| PHYSICOCHEMICAL PROPERTIES AND ANTIMICROBIAL ACTIVITY OF NEW SPIROCYCLIC THIENO[2,3-d]PYRIMIDIN-4(3H)-ONE DERIVATIVES |
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| Modesto de Candia, Claudia Altamura, Nunzio Denora, Saverio Cellamare, Manuel Nuzzolese, Danila De Vito, Leonid G. Voskressensky, Alexey V. Varlamov, Cosimo D. Altomare | 357-363 |
| SYNTHESIS OF NEW HETEROCYCLIC DEHYDROABIETYLAMINE DERIVATIVES AND THEIR BIOLOGICAL ACTIVITY |
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| Ксения С. Ковалева, Ольга И. Яровая, Андрей В. Шернюков, Владимир В. Зарубаев, Анна А. Штро, Яна Р. Оршанская, Нариман Ф. Салахутдинов | 364-370 |
| SYNTHESIS AND BIOLOGICAL ACTIVITY OF HETEROCYCLIC BORNEOL DERIVATIVES |
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| Anastasiya S. Sokolova, Olga I. Yarovaya, Anna A. Shtro, Marina S. Borisova, Ekaterina A. Morozova, Tatyana G. Tolstikova, Vladimir V. Zarubaev, Nariman F. Salakhutdinov | 371-377 |
Letters to the Editor
| (5S,7R)-5-Aryl-7-methyl-4,5,6,7-tetrahydro[1,2,4]triazolo[1,5-a]pyrimidin-7-ols as products of three-component condensation |
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| Sergey A. Komykhov, Andrey A. Bondarenko, Vladimir I. Musatov, Mikhail V. Diachkov, Nikolay Yu. Gorobets, Sergey M. Desenko | 378-380 |
Latvian Institute of Organic Synthesis - Aizkraukles iela, 21, Riga, LV-1006, Latvia - hgs@osi.lv