Vol 53, No 3 (2017)

Privileged heterocyclic scaffolds in chemical biology and drug discovery: synthesis and bioactivity

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Open Access Open Access  Restricted Access Subscription Access
2017 No. 3 (597) pp. 239–380

Table of Contents

Editorial

PRIVILEGED HETEROCYCLIC SCAFFOLDS IN CHEMICAL BIOLOGY AND DRUG DISCOVERY: SYNTHESIS AND BIOACTIVITY PDF
Cosimo D. Altomare 239

Review Articles

N-(HETERO)ARYL-2-IMIDAZOLINES: AN EMERGING PRIVILEGED MOTIF FOR CONTEMPORARY DRUG DESIGN PDF
Mikhail Krasavin 240-255
PREPARATION AND BIOLOGICAL PROPERTIES OF 2-THIO-CONTAINING PYRIMIDINES AND THEIR CONDENSED ANALOGS PDF
Oleksii Y. Voskoboynik, Oleksandra S. Kolomoets, Galina G. Berest, Inna S. Nosulenko, Yuliya V. Martynenko, Sergiy I. Kovalenko 256-273
HETEROCYCLES AS CLASSICAL AND NONCLASSICAL RING B ISOSTERS IN COMBRETASTATIN A-4 PDF
Nikolay A. Zefirov, Olga N. Zefirova 273-280
1,5-DIARYLPYRROLES AS POTENT ANTITUBERCULAR AND ANTI-INFLAMMATORY AGENTS PDF
Giulia Venditti, Giovanna Poce, Sara Consalvi, Mariangela Biava 281-291
2-(AZOLYL)ANILINES: METHODS OF SYNTHESIS, CYCLOCONDENSATIONS, AND BIOLOGICAL PROPERTIES PDF
Oleksii M. Antypenko, Sergiy V. Kholodnyak, Konstantin P. Schabelnyk, Lyudmyla M. Antypenko, Sergiy Ivanovich Kovalenko 292-309

Heterocycles in Focus

3,4-DIHYDROQUINOXALIN-2-ONES: RECENT ADVANCES IN SYNTHESIS AND BIOACTIVITIES PDF
Tone Kristoffersen, Jørn H. Hansen 310-312
SYNTHESIS OF INDOLIZINIUM SALTS PDF
Anna Ivanova, Pavel Arsenyan 313-315

Original Papers

EXPLORING THE INFLUENCE OF THE SUBSTITUENT AT POSITION 4 IN A SERIES OF 3,4-DIHYDROPYRIMIDIN-2(1H)-ONE A2B ADENOSINE RECEPTOR ANTAGONISTS PDF
Abel Crespo, Abdelaziz El Maatougui, Jhonny Azuaje, Luz Escalante, María Majellaro, María I. Loza, José Brea, María I. Cadavid, Hugo Gutiérrez-de-Terán, Eddy Sotelo 316-321
FUNCTIONALIZATION OF FOUR-MEMBERED CYCLIC SULFOXIMINES BY A CONVENIENT LITHIATION/TRAPPING SEQUENCE PDF
Arianna Tota, Flavio Fanelli, Aurelia Falcicchio, Renzo Luisi, Leonardo DEGENNARO 322-328
2-ARYLAZETINES AS LIGANDS FOR NICOTINIC ACETYLCHOLINE RECEPTORS PDF
Leonardo Degennaro, Marina Zenzola, Annunziatina Laurino, Maria Maddalena Cavalluzzi, Carlo Franchini, Solomon Habtemariam, Rosanna Matucci, Renzo Luisi, Giovanni Lentini 329-334
SYNTHESIS AND STRUCTURE OF DIHYDROBERBERINE NITROARYL DERIVATIVES – POTENTIAL LIGANDS FOR G-QUADRUPLEXES PDF (Russian)
Олег Н. Буров, Сергей В. Курбатов, Михаил Е. Клецкий, Александр Д. Загребаев, Игорь Е. Михайлов 335-340
INVESTIGATION ON THE SYNTHESIS OF NEW 3-[4-(ARYLALKOXY)PHENYLETHYL]-2-THIOXO-1,3-THIAZOLIDIN-4-ONES AND THEIR BIOLOGICAL EVALUATION AGAINST CANCER CELLS PDF
Camille D. Dago, Christelle N'ta Ambeu, Wacothon K. Coulibaly, Janat A. Mamyrbekova-Bekro, Rémy Le Guével, Anne Corlu, Jean-Pierre Bazureau 341-349
SYNTHESIS OF PHENYLPYRIDINE DERIVATIVES AND THEIR BIOLOGICAL EVALUATION TOWARD DIPEPTIDYL PEPTIDASE-4 PDF
Yan Zhu, Xiangguo Meng, Zhengyan Cai, Qun Hao, Weicheng Zhou 350-356
PHYSICOCHEMICAL PROPERTIES AND ANTIMICROBIAL ACTIVITY OF NEW SPIROCYCLIC THIENO[2,3-d]PYRIMIDIN-4(3H)-ONE DERIVATIVES PDF
Modesto de Candia, Claudia Altamura, Nunzio Denora, Saverio Cellamare, Manuel Nuzzolese, Danila De Vito, Leonid G. Voskressensky, Alexey V. Varlamov, Cosimo D. Altomare 357-363
SYNTHESIS OF NEW HETEROCYCLIC DEHYDROABIETYLAMINE DERIVATIVES AND THEIR BIOLOGICAL ACTIVITY PDF (Russian)
Ксения С. Ковалева, Ольга И. Яровая, Андрей В. Шернюков, Владимир В. Зарубаев, Анна А. Штро, Яна Р. Оршанская, Нариман Ф. Салахутдинов 364-370
SYNTHESIS AND BIOLOGICAL ACTIVITY OF HETEROCYCLIC BORNEOL DERIVATIVES PDF
Anastasiya S. Sokolova, Olga I. Yarovaya, Anna A. Shtro, Marina S. Borisova, Ekaterina A. Morozova, Tatyana G. Tolstikova, Vladimir V. Zarubaev, Nariman F. Salakhutdinov 371-377

Letters to the Editor

(5S,7R)-5-Aryl-7-methyl-4,5,6,7-tetrahydro[1,2,4]triazolo[1,5-a]pyrimidin-7-ols as products of three-component condensation PDF
Sergey A. Komykhov, Andrey A. Bondarenko, Vladimir I. Musatov, Mikhail V. Diachkov, Nikolay Yu. Gorobets, Sergey M. Desenko 378-380


 

 

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