

2016 No. 1 (583) pp. 1–70
Table of Contents
Heterocycles in Focus
SYNTHESIS OF 4H-THIAZINES |
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Aurelija Urbanaite, Inga Čikotienė | 1-3 |

NH-1,2,3-TRIAZOLES: SYNTHESIS AND REACTIONS WITH ELECTROPHILIC AGENTS |
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Василий A. Бакулев, Татьяна В. Березкина | 4-6 |

ALKYLIDENE AND ARYLIDENE MELDRUM'S ACIDS AS VERSATILE REAGENTS FOR THE SYNTHESIS OF HETEROCYCLES |
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Inese Mieriņa, Māra Jure | 7-9 |

NITROOLEFINS AS STARTING MATERIALS FOR 5-MEMBERED N-HETEROCYCLES |
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Inese Mieriņa, Māra Jure | 10-12 |

O,S-DISUBSTITUTED XANTHOGENATES IN HETEROCYCLIC SYNTHESIS |
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Петракис Н. Чаликиди | 13-14 |

Original Papers
MICROWAVE-ASSISTED ONE-POT SYNTHESIS OF PYRAZOLYL-SUBSTITUTED BENZOCHROMAN-4-ONE DERIVATIVES AND EVALUATION OF THEIR ANTICANCER ACTIVITY |
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Dongamanti Ashok, Kadiyala Padmavati, Bommidi Vijaya Lakshmi, Madderla Sarasija | 15-20 |

REDUCTION OF 5-(INDOL-3-YL)PYRROLIDIN-2-ONES |
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Андрей В. Садовой, Вита Н. Никитина, Виктор Б. Рыбаков, Константин А. Кочетков, Людмила А. Свиридова | 21-24 |

NEW N-MANNICH BASES OBTAINED FROM ISATIN AND PIPERAZINE DERIVATIVES: THE SYNTHESIS AND EVALUATION OF ANTIMICROBIAL ACTIVITY |
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Андрей В. Богданов, Альбина М. Вазыхова, Надежда Р. Хасиятуллина, Дмитрий Б. Криволапов, Алексей Б. Добрынин, Александра Д. Волошина, Владимир Ф. Миронов | 25-30 |

SOLVENT-FREE REGIOSELECTIVE SYNTHESIS OF NOVEL ISOXAZOLINE AND PYRAZOLINE N-SUBSTITUTED SACCHARIN DERIVATIVES UNDER MICROWAVE IRRADIATION |
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Aziza Saber, Mohsine Driowya, Soukaina Alaoui, Hamid Marzag, Luc Demange, Eleuterio Álvarez, Rachid Benhida, Khalid Bougrin | 31-40 |


SYNTHESIS OF N-ALKYLATED BENZO- AND PYRIDOTHIENOPYRROLO[1,2-a][1,4]DIAZEPIN-6-ONES ACTING AS ANTIDOTES AGAINST THE HERBICIDE 2,4-D |
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Татьяна А. Строганова, Владимир К. Василин, Геннадий Д. Крапивин, Владимир Д. Стрелков, Людмила В. Дядюченко | 45-51 |

ISOXAZOLO[4,3-e]INDAZOLE AS A NEW HETEROCYCLIC SYSTEM: DESIGN, SYNTHESIS, SPECTROSCOPIC CHARACTERIZATION, AND ANTIBACTERIAL ACTIVITY |
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Masoumeh Ghaemi, Mehdi Pordel | 52-57 |

SYNTHESIS OF 1-FUNCTIONALLY SUBSTITUTED DERIVATIVES OF DI- AND TETRAMETHYL- 3,4-DIHYDROBENZOFURO[3,2-g]- AND [2,3-h]ISOQUINOLINES |
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Татьяна С. Вшивкова, Алексей А. Горбунов, Ольга А. Майорова, Павел А. Слепухин, Максим Л. Исенов, Юрий В. Шкляев | 58-67 |

Letters to the Editor
THE FIRST SYNTHESIS OF 6-(PHENYLETHYNYL)-SUBSTITUTED TETRAHYDROAZOCINO[5,4-b]INDOLES |
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Леонид Г. Воскресенский, Александр А. Титов, Максим С. Кобзев, Реза Самавати, Роман С. Борисов, Лариса Н. Куликова, Алексей В. Варламов | 68-70 |

Chronicle
I Всероссийская молодежная школа-конференция "Успехи синтеза и комплексообразования" |
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Latvian Institute of Organic Synthesis - Aizkraukles iela, 21, Riga, LV-1006, Latvia - hgs@osi.lv