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Vol. 61 No. 11/12 (2025)
Vol. 61 No. 11/12 (2025)
2025 № 11/12 (701/702)
Published:
2026-05-15
Anniversaries and dates
PROFESSOR SOLOMON HILLER AT 111: A TIMELESS INSPIRATION
Review Articles
PYRROLOTRIAZOLES
Dietrich Moderhack
A AMINOURACILS IN THE SYNTHESIS OF HETEROCYCLES
Rogheyeh Hossein Nia, Manouchehr Mamaghani, Fatame Tavakoli, Elham Saberikhah, Zahra Taati
Heterocycles in Focus
PHOTO-/ELECTROCATALYTIC CYCLIZATION OF QUINOXALIN-2(1H)-ONES: ASSEMBLY OF HIGHLY FUNCTIONALIZED HETEROCYCLES
Xin Han, Linlin Shi, Xin-Qi Hao
Original Papers
EVALUATION OF CHOLINESTERASE INHIBITORY POTENTIAL OF N-FURAN-2-YLMETHYL- AND N-THIOPHENE-2-YLMETHYLBENZAMIDE AND SULFONAMIDE DERIVATIVES
Muhammed Serdar, Ziya Dağalan, Ece Oğuz, Pınar Güller, Bilal Nişancı, Mehmet Koca
UNSATURATED CARBOHYDRATES AS A SCAFFOLD FOR THE C–Si BOND CONSTRUCTION
Jevgeņija Lugiņina, Karīna Ņikitina, Vladislavs Kroškins, Vitālijs Rjabovs
A SYNTHESIS OF POLYFUNCTIONALLY SUBSTITUTED CARBO- AND HETEROCYCLIC COMPOUNDS BASED ON A REACTION OF ETHYL ARYLMETHYLIDENECYANOACETATE WITH ACETOACETIC ACID N-ARYLAMIDES
Anush Khachatryan, Anush Sargsyan, Katya Avagyan, Anahit Simonyan, Angin Zohrabyan, Henrik Panosyan, Alik Badasyan
A [Et3NH][HSO4]-CATALYZED EFFICIENT, GREEN, AND SOLVENT-FREE SYNTHESIS OF 2,4,6-TRIARYLPYRIDINES
Satish V. Akolkar, Mubarak H. Shaikh, Amol A. Nagargoje, Krishna V. Lathi, Dipti D. More, Mininath K. Bhalmode, Santosh B. Kamble, Bapurao B. Shingate
THE ROTATIONAL BARRIER AND THE SUBSTITUENT EFFECT ON RELATIVE STABILITY OF MONOSUBSTITUTED PYRIDINES AND PYRIMIDINES
Ali H. Yateem
DESIGN AND DISCOVERY OF COMPOUND DXS05 AS A HIGHLY POTENT GSPT1 MOLECULAR GLUE DEGRADER
Li Zhang, Ling Wang, Meijing Deng, Huiying Wu, Shuting Zou, Gang Li, Zonghui Ma, Chao Zhang, Na Liu, Xinshan Deng
ONE-POT REDUCTIVE AMINATION OF 2-AZIDOBENZALDEHYDES WITH ALIPHATIC AMINES, N-PROPARGYLATION AND INTRAMOLECULAR (3+2) CYCLOADDITION FOR THE SYNTHESIS OF N-SUBSTITUTED TRIAZOLOBENZODIAZEPINES
Wensheng Zhang, Wei Zheng, Xinling Du, Gaiyun Liu, Lvchen Wu
A FACILE PROTOCOL FOR THE DIRECT ARYLATION OF THIAZOLES UNDER COMBINED MICROWAVE AND ULTRASOUND IRRADIATION
Yanqiu Zhang, Zhiliang Zhang, Jiayi Wang, Yanqing Peng, Gonghua Song
EXPLORING FRIZZLED RECEPTOR MODULATION BY 2-(4-ISOPROPYLPHENYL)-5-NITROBENZOXAZOLE: A DUAL IN VITRO AND IN SILICO APPROACH
Burcu Baba, Çağla Z. Köprü, Erhan Oktay, Shoruq Ahmed Naji, Ayşegül Akbay, Ilkay Yildiz
OPTIMIZATION OF THE SYNTHESIS OF 2-(2-HYDROXYPHENYL)BENZAZOLE DYES IN POLYPHOSPHORIC ACID
Vanessa Cesar Ribas, Angelika von Schmude, Ingrid Maliszewski Paczkowski, Naira M. Balzaretti, Leandra Franciscato Campo
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